UCN-01（7-Hydroxystaurosporine；NSC 638850）是 staurosporine 的合成衍生物，对多种体外和体内癌症模型具有抗增殖活性。

Go 6983 是一种针对 PKCα、PKCβ、PKCγ 和 PKCδ 的泛 PKC 抑制剂，IC50 分别为 7 nM、7 nM、6 nM 和 10 nM。

TV 3279 is a novel ChE-MAI inhibitor , and the neuroprotective properties depend on their ability to induce the anti-apoptotic proteins PKC, Bcl-2, Bcl-x, and SOD, and to block the nuclear translocation of the pro-apoptotic enzyme glyceraldehyde phosphate dehydrogenase in PC-12 and neuroblastoma cells.